SCHEMBL6238480

SCHEMBL6238480

CCN=C=NCCCN(C)C.O=COCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
SIGMAR1 Q99720 1/20 0.37
LTA4H P09960 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
HRH1 P35367 2/20 0.34
EGFR P00533 2/20 0.34
MEN1 O00255 1/20 0.33
PSMD14 O00487 1/20 0.33
KMT2A Q03164 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27802330 0.79 CYP1A2 (0.48) CYP1A2CYP2D6KDM4EHRH1KMT2A
Hydrochloric Acid SCHEMBL28087409 0.78 CYP1A2 (0.47) CYP1A2CYP2D6KDM4EHRH1KMT2A
SCHEMBL888152 0.75 CYP1A2 (0.53) CYP1A2CYP2D6SIGMAR1MAOAMAOB
Dimethylformamide SCHEMBL28206616 0.75 CYP1A2 (0.79) CYP1A2CYP2D6
Formic Acid SCHEMBL27558615 0.75 CYP1A2 (0.79) CYP1A2CYP2D6KDM4EMEN1KMT2A
Trimethylammonium SCHEMBL19813147 0.74 TSHR (0.44) MAOAMAOBTAAR1
SCHEMBL1372 0.74 CYP1A2 (1.00) CYP1A2CYP2D6
SCHEMBL4798477 0.74 CYP1A2 (1.00) CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL1689433 0.74 CYP1A2 (0.51) CYP1A2CYP2D6SIGMAR1MAOAMAOB
Dimethylformamide SCHEMBL28206599 0.73 CYP1A2 (0.76) CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307203-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2005-08-17 EP disclosed
EP-1307203-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-05-07 EP disclosed
WO-2001070232-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-09-27 WO disclosed