SCHEMBL624412

SCHEMBL624412

NCC1CCN(c2nn3cc(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 18/20 0.45
MAPT P10636 1/20 0.39
PIK3CA P42336 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627411 0.89 MAP3K12 (0.47) MAP3K12MAPTPIK3CA
SCHEMBL625202 0.89 MAP3K12 (0.43) MAP3K12MAPT
SCHEMBL625621 0.89 MAP3K12 (0.46) MAP3K12MAPTPIK3CA
SCHEMBL627373 0.86 MAP3K12 (0.46) MAP3K12MAPTPIK3CA
SCHEMBL626464 0.86 MAPT (0.47) MAP3K12MAPTPIK3CA
SCHEMBL625228 0.86 MAP3K12 (0.46) MAP3K12PIK3CA
SCHEMBL626169 0.85 MAP3K12 (0.41) MAP3K12MAPTPIK3CA
SCHEMBL624411 0.85 PIK3CA (0.54) PIK3CA
SCHEMBL624389 0.84 MAP3K12 (0.43) MAP3K12PIK3CA
SCHEMBL626392 0.83 MAP3K12 (0.44) MAP3K12MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed