SCHEMBL6246335

SCHEMBL6246335

CN1CCN(C(=O)N=O)CC1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
HTR1A P08908 1/20 0.43
HTT P42858 1/20 0.39
HSD11B1 P28845 1/20 0.39
PHGDH O43175 1/20 0.39
MGLL Q99685 1/20 0.39
POLB P06746 2/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
MAPT P10636 1/20 0.37
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL735366 0.82 CYP1A2 (0.56) CYP1A2TDP1HTR1AHTTHSD11B1
SCHEMBL735365 0.82 CYP1A2 (0.56) CYP1A2TDP1HTR1AHTTHSD11B1
SCHEMBL2288243 0.80 CYP1A2 (0.54) CYP1A2TDP1HTR1AHTTHSD11B1
SCHEMBL5470776 0.73 CYP1A2 (0.65) CYP1A2TDP1HTR1AHTTHSD11B1
SCHEMBL33260 0.70 CYP1A2 (1.00) CYP1A2TDP1HTR1AHTTHSD11B1
SCHEMBL1965092 0.70 CYP1A2 (0.62) CYP1A2TDP1HTR1AHTTHSD11B1
SCHEMBL15531 0.70 TDP1 (0.62) CYP1A2TDP1HTR1AHTTHSD11B1
SCHEMBL13925516 0.70 CYP1A2 (1.00) CYP1A2TDP1HTR1AHTTHSD11B1
SCHEMBL4508546 0.70 TDP1 (0.62) CYP1A2TDP1HTR1AHTTHSD11B1
Hydrochloric Acid SCHEMBL15209250 0.70 CYP1A2 (0.62) CYP1A2TDP1HTR1AHTTHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017087667-A9 A SOLID STATE FORM OF PLADIENOLIDE PYRIDINE COMPOUNDS AND METHODS OF USE EISAI R&D MANAGEMENT CO., LTD. (JP) 2017-10-12 WO disclosed
WO-2005030237-A1 A PHARMACEUTICAL COMPOSITION COMPRISING CATHARANTHUS ROSEAUS, (VINCA ROSEA), ITS PREPARATION AND USE THEREOF SEÑOR RAFAEL PHIL. INC. (PH) 2005-04-07 WO disclosed