SCHEMBL6252961

SCHEMBL6252961

N#Cc1c(N)nc2sc(C(N)=O)c(N)c2c1-c1cccnc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.70
HSP90AB1 P08238 1/20 0.62
ALDH1A1 P00352 4/20 0.61
EEF2K O00418 1/20 0.60
LIMK1 P53667 1/20 0.54
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
MAPK1 P28482 3/20 0.53
NPSR1 Q6W5P4 2/20 0.53
HPGD P15428 1/20 0.53
PDE4A P27815 1/20 0.52
PDE4B Q07343 1/20 0.52
PDE4C Q08493 1/20 0.52
PDE4D Q08499 1/20 0.52
KDM4E B2RXH2 4/20 0.51
HSD17B10 Q99714 3/20 0.51
HTT P42858 2/20 0.51
MAPT P10636 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
RXFP1 Q9HBX9 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1775711 0.88 BRAF (0.81) BRAFHSP90AB1ALDH1A1LIMK1MEN1
SCHEMBL6258124 0.87 BRAF (0.79) BRAFHSP90AB1ALDH1A1EEF2KMEN1
SCHEMBL1775859 0.83 BRAF (0.70) BRAFHSP90AB1ALDH1A1EEF2KMEN1
SCHEMBL1776805 0.83 BRAF (0.77) BRAFHSP90AB1ALDH1A1EEF2KLIMK1
SCHEMBL6257937 0.82 BRAF (0.83) BRAFHSP90AB1ALDH1A1EEF2KMEN1
SCHEMBL1776085 0.82 BRAF (1.00) BRAFHSP90AB1ALDH1A1EEF2KLIMK1
SCHEMBL6253458 0.82 BRAF (0.69) BRAFHSP90AB1ALDH1A1EEF2KMEN1
SCHEMBL6256957 0.82 BRAF (0.69) BRAFHSP90AB1ALDH1A1EEF2KMEN1
SCHEMBL6255310 0.81 BRAF (0.74) BRAFHSP90AB1ALDH1A1EEF2KMEN1
SCHEMBL6254816 0.81 BRAF (0.81) BRAFHSP90AB1ALDH1A1EEF2KMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005058315-A1 NOVEL HETEROCYCLIC COMPOUNDS AS IKK2 INHIBITORS WITH ANTI-HBV ACTIVITY RIBAPHARM, INC. (US) 2005-06-30 WO disclosed