SCHEMBL6253145

SCHEMBL6253145

O=C(O)c1ccc(-c2ccc(C(=O)O)cc2Cl)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 4/20 0.72
TSHR P16473 3/20 0.61
ADH5 P11766 2/20 0.60
RXRA P19793 1/20 0.55
RXRB P28702 1/20 0.55
TNKS2 Q9H2K2 1/20 0.55
ALOX15 P16050 1/20 0.50
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
CRHBP P24387 1/20 0.49
RAB9A P51151 1/20 0.49
CRHR2 Q13324 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HSD17B1 P14061 1/20 0.49
HSD17B2 P37059 1/20 0.49
ADRB1 P08588 1/20 0.48
ADRB3 P13945 1/20 0.48
TP53 P04637 1/20 0.48
FOLH1 Q04609 1/20 0.47
TTR P02766 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9812960 0.98 SRD5A2 (0.70) SRD5A2TSHRADH5RXRARXRB
SCHEMBL23484575 0.92 SRD5A2 (0.73) SRD5A2TSHRADH5RXRARXRB
SCHEMBL8082912 0.91 SRD5A2 (0.61) SRD5A2TSHRADH5RXRARXRB
SCHEMBL2044221 0.90 SRD5A2 (0.60) SRD5A2TSHRADH5RXRARXRB
SCHEMBL444367 0.89 SRD5A2 (0.90) SRD5A2TSHRADH5RXRARXRB
SCHEMBL2769863 0.87 TSHR (0.71) SRD5A2TSHRADH5RXRARXRB
SCHEMBL10717595 0.87 SRD5A2 (0.66) SRD5A2ADH5RXRARXRBHSD17B1
SCHEMBL3741905 0.85 SRD5A2 (0.64) SRD5A2TSHRADH5RXRARXRB
SCHEMBL8144296 0.85 SRD5A2 (0.64) SRD5A2TSHRADH5RXRARXRB
SCHEMBL3758566 0.85 SRD5A2 (0.64) SRD5A2TSHRADH5RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569954-A1 CYANOMETHYL DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-09-07 EP disclosed
WO-2004052921-A1 CYANOMETHYL DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-06-24 WO disclosed
EP-0539243-B1 Process for introducing a carboxyl group to an aromatic carboxylic acid or a derivative thereof HIRAI HIDEFUMI (JP) 1996-01-24 EP disclosed
US-5319134-A Process for introducing a carboxyl group to an aromatic carboxylic acid or a derivative thereof HIDEFUMI HIRAI (JP) 1994-06-07 US disclosed
EP-0539243-A2 Process for introducing a carboxyl group to an aromatic carboxylic acid or a derivative thereof Hirai, Hidefumi (JP) 1993-04-28 EP disclosed