SCHEMBL625645

SCHEMBL625645

Nc1ncc(-c2cnc3sc(N4CCN5CCNCC5C4)nn23)cc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.47
MAP3K12 Q12852 6/20 0.38
KCNH2 Q12809 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625646 0.86 MAP3K12 (0.41) MAP3K12
SCHEMBL624388 0.84 PIK3CA (0.55) PIK3CAMAP3K12KCNH2
SCHEMBL626160 0.82 PIK3CA (0.50) PIK3CAMAP3K12KCNH2
SCHEMBL625227 0.80 PIK3CA (0.55) PIK3CAMAP3K12KCNH2
SCHEMBL626245 0.80 PIK3CA (0.46) PIK3CAMAP3K12KCNH2
SCHEMBL625018 0.78 PIK3CA (0.51) PIK3CAKCNH2
SCHEMBL627410 0.78 PIK3CA (0.57) PIK3CAKCNH2
SCHEMBL624438 0.78 PIK3CA (0.50) PIK3CAKCNH2
SCHEMBL625620 0.77 PIK3CA (0.56) PIK3CAKCNH2
SCHEMBL625458 0.77 PIK3CA (0.51) PIK3CAMAP3K12KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed