SCHEMBL625702

SCHEMBL625702

CS(=O)(=O)N1CC2(CCCN(c3nn4c(-c5cnc(N)c(C(F)(F)F)c5)cnc4s3)C2)C1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 9/20 0.50
MAP3K12 Q12852 1/20 0.41
EIF2AK4 Q9P2K8 1/20 0.41
HASPIN Q8TF76 4/20 0.40
KCNH2 Q12809 3/20 0.38
FLT3 P36888 2/20 0.38
PIM1 P11309 2/20 0.38
KIT P10721 1/20 0.38
CDK7 P50613 1/20 0.38
PIM3 Q86V86 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626242 0.89 PIK3CA (0.52) PIK3CAMAP3K12HASPINKCNH2FLT3
SCHEMBL625703 0.87 MAP3K12 (0.44) PIK3CAMAP3K12EIF2AK4
SCHEMBL626122 0.83 PIK3CA (0.45) PIK3CAEIF2AK4HASPINKCNH2FLT3
SCHEMBL626461 0.83 PIK3CA (0.47) PIK3CAHASPINKCNH2FLT3PIM1
SCHEMBL626619 0.82 PIK3CA (0.55) PIK3CAMAP3K12HASPINKCNH2
SCHEMBL626262 0.79 PIK3CA (0.54) PIK3CAMAP3K12HASPINKCNH2FLT3
SCHEMBL626160 0.79 PIK3CA (0.50) PIK3CAMAP3K12KCNH2
SCHEMBL625458 0.78 PIK3CA (0.51) PIK3CAMAP3K12HASPINKCNH2FLT3
SCHEMBL627019 0.78 PIK3CA (0.47) PIK3CAMAP3K12HASPINKCNH2FLT3
SCHEMBL624869 0.77 PIK3CA (0.52) PIK3CAMAP3K12HASPINKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed