SCHEMBL6259747

SCHEMBL6259747

CN(Cc1cc(Cl)cc(Cl)c1)C(=O)C1CN(C(=O)O)CCN1c1ccc(F)cc1F

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.45
CCR1 P32246 4/20 0.40
HTT P42858 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
GRM5 P41594 1/20 0.36
NPC1 O15118 1/20 0.36
TACR3 P29371 1/20 0.36
P2RX7 Q99572 1/20 0.35
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PABPC1 P11940 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6257518 0.92 TACR1 (0.54) TACR1CCR1HTTKDM4EMEN1
SCHEMBL6263440 0.88 CCR1 (0.43) TACR1CCR1HTTKDM4EMEN1
SCHEMBL6259791 0.88 CCR1 (0.39) TACR1CCR1HTTKDM4EMEN1
SCHEMBL5394686 0.87 TACR1 (0.44) TACR1SMN1; SMN2
SCHEMBL6261488 0.87 TACR1 (0.61) TACR1
SCHEMBL6264225 0.83 TACR1 (0.51) TACR1CCR1TACR3P2RX7
SCHEMBL6258643 0.83 TACR1 (0.54) TACR1CCR1
SCHEMBL5389958 0.80 TACR1 (0.52) TACR1
SCHEMBL6261284 0.80 CCR1 (0.46) TACR1CCR1
SCHEMBL6262695 0.79 TACR1 (0.47) TACR1CCR1P2RX7SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1423117-B1 2-SUBSTITUTED 1-ARYLPIPERAZINES AS TACHYKININ ANTAGONISTS AND/OR SEROTONIN REUPTAKE INHIBITORS GLAXO GROUP LTD (GB) 2005-10-19 EP disclosed