SCHEMBL627372

SCHEMBL627372

COC1CCN(c2nn3c(-c4cnc(N)c(C(F)(F)F)c4)cnc3s2)CC1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.57
KCNH2 Q12809 7/20 0.45
HASPIN Q8TF76 3/20 0.44
FLT3 P36888 2/20 0.44
KIT P10721 1/20 0.44
PIM1 P11309 1/20 0.44
CDK7 P50613 1/20 0.44
PIM3 Q86V86 1/20 0.44
PIM2 Q9P1W9 1/20 0.44
MAP3K12 Q12852 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627410 0.88 PIK3CA (0.57) PIK3CAKCNH2HASPINFLT3KIT
SCHEMBL625620 0.87 PIK3CA (0.56) PIK3CAKCNH2HASPINFLT3KIT
SCHEMBL625746 0.87 PIK3CA (0.54) PIK3CAKCNH2HASPINFLT3KIT
SCHEMBL624411 0.85 PIK3CA (0.54) PIK3CAKCNH2HASPINFLT3KIT
SCHEMBL627373 0.85 MAP3K12 (0.46) PIK3CAMAP3K12
SCHEMBL626463 0.85 PIK3CA (0.53) PIK3CAKCNH2
SCHEMBL625227 0.84 PIK3CA (0.55) PIK3CAKCNH2HASPINFLT3KIT
SCHEMBL624388 0.83 PIK3CA (0.55) PIK3CAKCNH2HASPINFLT3KIT
SCHEMBL624967 0.83 PIK3CA (0.55) PIK3CAKCNH2HASPINFLT3KIT
SCHEMBL627785 0.82 PIK3CA (0.56) PIK3CAPIM1MAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed