SCHEMBL6276773

SCHEMBL6276773

CN(CCF)CCC1=C(Cc2cnccn2)c2ccccc2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 18/20 1.00
CYP2D6 P10635 17/20 1.00
CYP3A4 P08684 3/20 0.82
KCNH2 Q12809 5/20 0.80
CHRM1 P11229 3/20 0.80
HTR2A P28223 1/20 0.80
CHRM2 P08172 2/20 0.60
CHRM4 P08173 2/20 0.60
CHRM5 P08912 2/20 0.60
CHRM3 P20309 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6278779 0.89 HRH1 (1.00) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6270302 0.78 HRH1 (0.80) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6278192 0.77 HRH1 (1.00) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6272080 0.76 CYP2D6 (1.00) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6266110 0.74 HRH1 (1.00) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6415321 0.72 HRH1 (0.82) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6279585 0.67 HRH1 (0.81) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6270161 0.67 HRH1 (0.84) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6279444 0.67 HRH1 (0.81) HRH1CYP2D6CYP3A4KCNH2CHRM1
SCHEMBL6418786 0.67 HRH1 (0.80) HRH1CYP2D6CYP3A4KCNH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005097093-A1 SLEEP INDUCING COMPOUNDS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2005-10-20 WO disclosed