SCHEMBL6276896

SCHEMBL6276896

CC(C)C1OC1c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 11/20 0.61
TSHR P16473 2/20 0.39
SLC6A2 P23975 1/20 0.34
ADRA1A P35348 1/20 0.34
HTR2B P41595 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8508730 0.84 EPHX1 (0.59) EPHX1TSHRSLC6A2ADRA1AHTR2B
SCHEMBL28357174 0.82 EPHX1 (0.68) EPHX1TSHR
SCHEMBL28353670 0.82 EPHX1 (0.68) EPHX1TSHR
SCHEMBL28353669 0.82 EPHX1 (0.68) EPHX1TSHR
SCHEMBL4113792 0.82 EPHX1 (0.68) EPHX1TSHR
SCHEMBL28353827 0.82 EPHX1 (0.68) EPHX1TSHR
SCHEMBL28357172 0.82 EPHX1 (0.68) EPHX1TSHR
SCHEMBL13773134 0.79 EPHX1 (0.44) EPHX1TSHR
SCHEMBL20634564 0.79 EPHX1 (0.44) EPHX1TSHR
SCHEMBL13773136 0.79 EPHX1 (0.44) EPHX1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11739074-B2 Ras inhibitors Revolution Medicines, Inc. (US) 2023-08-29 US disclosed
US-11739074-B2 Ras inhibitors Revolution Medicines, Inc. (US) 2023-08-29 US disclosed
US-20230233569-A1 METHODS FOR DELAYING, PREVENTING, AND TREATING ACQUIRED RESISTANCE TO RAS INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION, AS AGENT 2023-07-27 US disclosed
US-20210130326-A1 RAS INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION, AS AGENT 2021-05-06 US disclosed
EP-1317460-A4 COMPOUNDS CONTAINING OXAZOLIDINONE MOIETY AND USES THEREOF UNIV COLORADO STATE RES FOUND (US) 2005-04-20 EP disclosed
EP-1317460-A1 COMPOUNDS CONTAINING OXAZOLIDINONE MOIETY AND USES THEREOF COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2003-06-11 EP disclosed
EP-0724569-B1 PROCESS FOR THE PREPARATION OF AN OXIRANE, AZIRIDINE OR CYCLOPROPANE AVECIA LTD (GB) 2003-03-12 EP disclosed
WO-2002018391-A1 COMPOUNDS CONTAINING OXAZOLIDINONE MOIETY AND USES THEREOF COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2002-03-07 WO disclosed
US-5703246-A REACTING AN ORGANOMETALLIC COMPOUND WITH ORGANOSULFUR COMPOUND ZENECA LIMITED (GB) 1997-12-30 US disclosed
EP-0724569-A1 PROCESS FOR THE PREPARATION OF AN OXIRANE, AZIRIDINE OR CYCLOPROPANE ZENECA LIMITED (GB) 1996-08-07 EP disclosed
WO-1995011230-A1 PROCESS FOR THE PREPARATION OF AN OXIRANE, AZIRIDINE OR CYCLOPROPANE ZENECA LIMITED (GB) 1995-04-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11739074-B2 Ras inhibitors KRAS, NRAS, HRAS EPHX1 2296/4885TSHR 3396/4885SLC6A2 4824/4885
US-20210130326-A1 RAS INHIBITORS KRAS, NRAS, HRAS EPHX1 2887/4885TSHR 3332/4885SLC6A2 4833/4885
US-20230233569-A1 METHODS FOR DELAYING, PREVENTING, AND TREATING ACQUIRED RESISTANCE TO RAS INHIBITORS KRAS, HRAS, MTOR EPHX1 3640/4885TSHR 4120/4885SLC6A2 4621/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.