SCHEMBL6281985

SCHEMBL6281985

COc1c(C(=O)Cl)c(-c2ccccc2)nn1-c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
ALDH1A1 P00352 5/20 0.48
MPO P05164 1/20 0.46
SRC P12931 1/20 0.44
BRAF P15056 1/20 0.44
KDR P35968 1/20 0.44
MAPT P10636 3/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TP53 P04637 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6270116 0.89 MEN1 (0.67) MEN1KMT2AALDH1A1MPOSRC
Hydrochloric Acid SCHEMBL6281990 0.87 MEN1 (0.65) MEN1KMT2AALDH1A1MPOSRC
SCHEMBL6267877 0.81 MEN1 (0.78) MEN1KMT2AALDH1A1SRCBRAF
SCHEMBL11476853 0.74 CYP1A2 (0.61) MEN1KMT2AMPOMAPTCYP2C9
SCHEMBL14553211 0.73 MEN1 (0.75) MEN1KMT2AALDH1A1MAPTCYP2C9
SCHEMBL14132507 0.73 MEN1 (1.00) MEN1KMT2AALDH1A1SRCBRAF
SCHEMBL1553100 0.72 MEN1 (1.00) MEN1KMT2AALDH1A1SRCBRAF
SCHEMBL6269787 0.71 MEN1 (0.58) MEN1KMT2AALDH1A1SRCBRAF
SCHEMBL14133375 0.70 MEN1 (0.69) MEN1KMT2AALDH1A1SRCBRAF
SCHEMBL4494401 0.70 CYP2C9 (0.69) MEN1KMT2AALDH1A1SRCBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005061462-A2 DIARYL PYRAZOLE DERIVATIVES AND THEIR USE AS NEUROKININ-3 RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2005-07-07 WO disclosed