SCHEMBL6288933

SCHEMBL6288933

CCN1CCN(c2nc(-c3ccc(-c4cccc(OC)c4)cc3)cc3ccccc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.49
CYP1A2 P05177 4/20 0.49
CYP3A4 P08684 4/20 0.49
USP2 O75604 3/20 0.49
CLK4 Q9HAZ1 3/20 0.49
TSHR P16473 2/20 0.49
MAPK1 P28482 2/20 0.49
ABCG2 Q9UNQ0 1/20 0.47
TP53 P04637 1/20 0.46
FGFR1 P11362 1/20 0.45
LMNA P02545 3/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP2C19 P33261 2/20 0.44
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
HIF1A Q16665 1/20 0.44
HPGD P15428 2/20 0.44
MAPT P10636 2/20 0.44
HSD17B10 Q99714 2/20 0.44
KDR P35968 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768407 0.95 TSHR (0.52) CYP2D6CYP1A2CYP3A4USP2CLK4
Hydrochloric Acid SCHEMBL4764011 0.94 TSHR (0.51) CYP2D6CYP1A2CYP3A4USP2CLK4
SCHEMBL4763566 0.90 HRH3 (0.48) CYP1A2LMNAALDH1A1CYP2C19HPGD
Hydrochloric Acid SCHEMBL4770729 0.89 HRH3 (0.47) CYP1A2TSHRLMNAALDH1A1CYP2C19
SCHEMBL4774077 0.88 SMN1; SMN2 (0.46) CYP2D6CYP1A2CYP3A4USP2CLK4
Hydrochloric Acid SCHEMBL4768944 0.87 SMN1; SMN2 (0.45) CYP2D6CYP1A2CYP3A4USP2CLK4
SCHEMBL4768596 0.86 SMN1; SMN2 (0.46) LMNAMAPTKMT2ASMN1; SMN2MEN1
Hydrochloric Acid SCHEMBL4766731 0.85 KMT2A (0.45) LMNAALDH1A1HPGDMAPTKMT2A
Hydrochloric Acid SCHEMBL6288704 0.85 KMT2A (0.45) LMNAALDH1A1HPGDMAPTKMT2A
SCHEMBL4767067 0.85 CYP2D6 (0.47) CYP2D6CYP1A2CYP3A4USP2CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6875761-B2 Certain 1,3-disubstituted isoquinoline derivatives EISAI CO., LTD. (JP) 2005-04-05 US disclosed