SCHEMBL629373

SCHEMBL629373

CC(=O)Nc1ccc(N2C(=O)N(CCCCCCCCCSCCCC(F)(F)C(F)(F)F)C(C)(C)C2=O)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.49
PGR P06401 1/20 0.49
HDAC1 Q13547 4/20 0.42
IGF1R P08069 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL891215 0.90 AR (0.46) ARPGRHDAC1
SCHEMBL629186 0.90 AR (0.45) ARPGR
SCHEMBL633694 0.89 AR (0.59) ARPGRHDAC1
SCHEMBL629084 0.87 AR (0.47) ARPGRHDAC1
SCHEMBL629322 0.85 AR (0.52) ARPGR
SCHEMBL629676 0.85 AR (0.50) ARPGRHDAC1
SCHEMBL629452 0.82 AR (0.50) ARPGR
SCHEMBL629766 0.82 AR (0.50) ARPGR
SCHEMBL630118 0.82 AR (0.50) ARPGR
SCHEMBL630258 0.82 AR (0.50) ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8710091-B2 Imidazolidine-2,4-dione derivatives, and use thereof as a cancer drug IPSEN PHARMA S.A.S. (FR) 2014-04-29 US disclosed
EP-2419410-B1 IMIDAZOLIDINE-2,4-DIONE DERIVATIVES, AND USE THEREOF AS A CANCER DRUG IPSEN PHARMA SAS (FR) 2013-03-06 EP disclosed
EP-2419410-A1 IMIDAZOLIDINE-2,4-DIONE DERIVATIVES, AND USE THEREOF AS A CANCER DRUG IPSEN PHARMA S.A.S. (FR) 2012-02-22 EP disclosed
WO-2010119193-A1 IMIDAZOLIDINE-2,4-DIONE DERIVATIVES, AND USE THEREOF AS A CANCER DRUG IPSEN PHARMA S.A.S. (FR) 2010-10-21 WO disclosed