SCHEMBL6299787

SCHEMBL6299787

COc1c(NC(=O)Nc2ccc(Oc3ccnc(N(C)CCN(C)C)c3)c3ccccc23)cc(C(C)(C)C)cc1NS(C)(=O)=O

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SRC P12931 14/20 0.70
SYK P43405 14/20 0.70
MAPK14 Q16539 12/20 0.70
GSK3A P49840 12/20 0.66
LCK P06239 2/20 0.64
CXCL8 P10145 2/20 0.61
TNF P01375 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6547053 0.90 SRC (0.71) SRCSYKMAPK14GSK3ALCK
SCHEMBL6545985 0.88 GSK3A (0.68) SRCSYKMAPK14GSK3ALCK
SCHEMBL6298580 0.87 GSK3A (0.69) SRCSYKMAPK14GSK3ACXCL8
SCHEMBL17659974 0.86 GSK3A (0.74) SRCSYKMAPK14GSK3ALCK
SCHEMBL6546000 0.86 GSK3A (0.74) SRCSYKMAPK14GSK3ALCK
SCHEMBL6546013 0.85 GSK3A (0.69) SRCSYKMAPK14GSK3ALCK
SCHEMBL18461774 0.85 GSK3A (0.73) SRCSYKMAPK14GSK3ALCK
SCHEMBL16143036 0.85 GSK3A (0.75) SRCSYKMAPK14GSK3ALCK
SCHEMBL17665876 0.85 GSK3A (0.73) SRCSYKMAPK14GSK3ALCK
SCHEMBL16106281 0.85 GSK3A (0.73) SRCSYKMAPK14GSK3ALCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6852717-B2 Compounds useful as anti-inflammatory agents BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-02-08 US disclosed