SCHEMBL6302902

SCHEMBL6302902

CC1Oc2ccc(CNCc3cccc(CNCc4ccc(Cl)cc4Cl)c3)cc2NC1=O

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.68
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDR P35968 1/20 0.40
HSD17B10 Q99714 1/20 0.39
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000465 0.96 PARP1 (0.67) PARP1TP53POLBSMN1; SMN2KDR
SCHEMBL6305046 0.90 PARP1 (0.77) PARP1TP53POLBSMN1; SMN2KDR
SCHEMBL6996295 0.88 PARP1 (0.78) PARP1TP53POLBSMN1; SMN2KDR
SCHEMBL6305288 0.87 PARP1 (0.88) PARP1TP53POLBSMN1; SMN2HSD17B10
SCHEMBL6304625 0.86 PARP1 (0.75) PARP1TP53POLBSMN1; SMN2KDR
SCHEMBL6992288 0.86 PARP1 (0.75) PARP1TP53POLBSMN1; SMN2ALDH1A1
SCHEMBL6999731 0.85 PARP1 (0.80) PARP1TP53POLBSMN1; SMN2HSD17B10
SCHEMBL6310170 0.84 PARP1 (0.95) PARP1TP53POLBSMN1; SMN2HSD17B10
SCHEMBL6999765 0.84 PARP1 (0.67) PARP1TP53POLBSMN1; SMN2KDR
SCHEMBL6309373 0.82 PARP1 (0.76) PARP1TP53POLBSMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6841550-B1 Benzoxazine and benzothiazine derivatives and their use in medicines SCHERING AKTIENGESELLSCHAFT (DE) 2005-01-11 US disclosed
EP-1114037-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES SCHERING AG (DE) 2004-05-12 EP disclosed