SCHEMBL6306583

SCHEMBL6306583

CC(C)C1Nc2ccccc2N(C)C(=O)C1NC(=O)[C@H](C)N

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
XIAP P98170 4/20 0.43
PSEN1 P49768 8/20 0.40
PSEN2 P49810 8/20 0.40
APH1B Q8WW43 8/20 0.40
NCSTN Q92542 8/20 0.40
APH1A Q96BI3 8/20 0.40
PSENEN Q9NZ42 8/20 0.40
CCKBR P32239 2/20 0.37
EGFR P00533 1/20 0.37
BRD4 O60885 1/20 0.36
KCNH2 Q12809 1/20 0.35
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6312860 0.99 XIAP (0.42) XIAPPSEN1PSEN2APH1BNCSTN
SCHEMBL6306461 0.85 BRD4 (0.42) XIAPPSEN1PSEN2APH1BNCSTN
SCHEMBL6308009 0.85 MEN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
Hydrochloric Acid SCHEMBL6312630 0.84 NOTCH1 (0.37) XIAPPSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL6305883 0.84 BRD4 (0.41) XIAPPSEN1PSEN2APH1BNCSTN
SCHEMBL6305563 0.80 SCN9A (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6912415 0.75 PSEN1 (0.56) XIAPPSEN1PSEN2APH1BNCSTN
SCHEMBL6305912 0.75 BRD4 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
Hydrochloric Acid SCHEMBL4411847 0.74 PSEN1 (0.55) XIAPPSEN1PSEN2APH1BNCSTN
SCHEMBL6300489 0.72 SCN9A (0.52) XIAPPSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6958330-B1 Polycyclic α-amino-ε-caprolactams and related compounds ELAN PHARMACEUTICALS, INC. (US) 2005-10-25 US disclosed