SCHEMBL6307600

SCHEMBL6307600

CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)NN1C(=O)C(CCCCc2ccccc2)c2ccccc2-c2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.42
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
ATM Q13315 1/20 0.41
CA2 P00918 1/20 0.41
CCKAR P32238 3/20 0.40
CCKBR P32239 3/20 0.40
GLS O94925 1/20 0.38
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
CASP3 P42574 1/20 0.37
APP P05067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6305076 0.92 SCN9A (0.43) SCN9AKMT2AATMCCKARCCKBR
SCHEMBL6309257 0.90 MEN1 (0.37) SCN9AKMT2AMEN1ATMCA2
SCHEMBL6307634 0.84 KMT2A (0.42) SCN9AKMT2AMEN1ATMCA2
SCHEMBL4424746 0.82 SCN9A (0.39) SCN9AKMT2AMEN1ATMCA2
SCHEMBL7568374 0.82 SCN9A (0.39) SCN9AKMT2AMEN1ATMCA2
SCHEMBL4418511 0.82 SCN9A (0.39) SCN9AKMT2AMEN1ATMCA2
SCHEMBL6307916 0.82 PSEN1 (0.41)
SCHEMBL6307499 0.81 PSEN1 (0.42) KMT2A
Hydrochloric Acid SCHEMBL4413409 0.81 PSEN1 (0.40)
Hydrochloric Acid SCHEMBL4411799 0.81 PSEN1 (0.41) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042298-A1 POLYCYCLIC ALPHA-AMINO-EPSILON-CAPROLACTAMS AND RELATED COMPOUNDS Elan Pharmaceuticals, Inc. (US) 2000-10-11 EP claimed
WO-1999032453-A1 POLYCYCLIC α-AMINO-⊂-CAPROLACTAMS AND RELATED COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 1999-07-01 WO claimed
US-6958330-B1 Polycyclic α-amino-ε-caprolactams and related compounds ELAN PHARMACEUTICALS, INC. (US) 2005-10-25 US disclosed
EP-1042298-A1 POLYCYCLIC ALPHA-AMINO-EPSILON-CAPROLACTAMS AND RELATED COMPOUNDS Elan Pharmaceuticals, Inc. (US) 2000-10-11 EP disclosed
WO-1999032453-A1 POLYCYCLIC α-AMINO-⊂-CAPROLACTAMS AND RELATED COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 1999-07-01 WO disclosed