SCHEMBL6326412

SCHEMBL6326412

O=C(CCc1nc(-c2ccc(F)cc2)no1)NCCCCNc1n[nH]c(=O)c2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.51
LMNA P02545 4/20 0.51
USP2 O75604 2/20 0.51
HPGD P15428 2/20 0.51
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
GAA P10253 5/20 0.49
HTT P42858 3/20 0.48
HDAC1 Q13547 2/20 0.47
HDAC2 Q92769 2/20 0.47
HDAC8 Q9BY41 1/20 0.47
CNR2 P34972 4/20 0.47
CNR1 P21554 1/20 0.46
ALDH1A1 P00352 3/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6326111 0.98 TSHR (0.51) TSHRLMNAUSP2HPGDCYP1A2
SCHEMBL6332518 0.96 HDAC1 (0.51) TSHRLMNAUSP2HPGDCYP1A2
SCHEMBL6334127 0.95 CYP1A2 (0.52) TSHRLMNAUSP2HPGDCYP1A2
SCHEMBL6325850 0.94 HDAC1 (0.51) TSHRLMNAUSP2HPGDCYP1A2
SCHEMBL6324028 0.93 HPGD (0.59) TSHRLMNAUSP2HPGDCYP1A2
SCHEMBL6327228 0.92 TSHR (0.58) TSHRLMNAUSP2HPGDCYP1A2
SCHEMBL6333112 0.92 TSHR (0.51) TSHRLMNAUSP2HPGDCYP1A2
SCHEMBL6327904 0.91 HPGD (0.59) TSHRLMNAUSP2HPGDCYP1A2
SCHEMBL6325569 0.91 HDAC1 (0.49) TSHRLMNAHPGDCYP1A2CYP2D6
SCHEMBL6328284 0.91 HPGD (0.52) TSHRLMNAUSP2HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924284-B2 PARP inhibitors ICOS CORPORATION (US) 2005-08-02 US disclosed