SCHEMBL6327072

SCHEMBL6327072

Cc1[nH]c(C=C2C(=O)Nc3cccc(-c4ccc(Cl)cc4)c32)c(C)c1CCC(=O)N1C[C@H](C)N[C@@H](C)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.50
FGFR1 P11362 15/20 0.50
PDGFRB P09619 14/20 0.50
RET P07949 3/20 0.50
FLT3 P36888 3/20 0.50
CHEK1 O14757 3/20 0.50
AURKA O14965 2/20 0.50
FLT1 P17948 2/20 0.50
MAP4K2 Q12851 2/20 0.50
STK3 Q13188 2/20 0.50
AURKB Q96GD4 2/20 0.50
ALK Q9UM73 2/20 0.50
GAK O14976 1/20 0.50
RPS6KA5 O75582 1/20 0.50
RPS6KA4 O75676 1/20 0.50
LATS1 O95835 1/20 0.50
CSNK2A2 P19784 1/20 0.50
MAP2K2 P36507 1/20 0.50
ZAP70 P43403 1/20 0.50
MAP2K1 Q02750 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6324365 1.00 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6327078 1.00 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6327070 1.00 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6324346 1.00 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6324350 1.00 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6330101 0.92 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6322670 0.92 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6330099 0.92 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6322677 0.92 KDR (0.50) KDRFGFR1PDGFRBRETFLT3
SCHEMBL6322659 0.92 KDR (0.50) KDRFGFR1PDGFRBRETFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677368-B2 4-aryl substituted indolinones SUGEN, INC. 2004-01-13 US claimed
US-6861418-B2 4-aryl substituted indolinones SUGEN, INC. (US) 2005-03-01 US disclosed
US-6677368-B2 4-aryl substituted indolinones SUGEN, INC. 2004-01-13 US disclosed