SCHEMBL6327593

SCHEMBL6327593

CC(C)C(CN1CCC(Cc2ccc(Cl)c(Cl)c2)CC1)Nc1nc2ccccc2o1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 4/20 0.52
SSTR5 P35346 14/20 0.46
HRH1 P35367 3/20 0.46
HTR2B P41595 2/20 0.46
OPRK1 P41145 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6327587 1.00 CCR3 (0.52) CCR3SSTR5HRH1HTR2BOPRK1
SCHEMBL6327582 1.00 CCR3 (0.52) CCR3SSTR5HRH1HTR2BOPRK1
SCHEMBL6331932 0.91 SSTR5 (0.47) CCR3SSTR5HRH1HTR2BOPRK1
SCHEMBL6326070 0.90 CCR3 (0.51) CCR3SSTR5HRH1HTR2B
SCHEMBL6326066 0.90 CCR3 (0.51) CCR3SSTR5HRH1HTR2B
SCHEMBL6326064 0.90 CCR3 (0.51) CCR3SSTR5HRH1HTR2B
SCHEMBL6325867 0.90 CCR3 (0.57) CCR3SSTR5HRH1HTR2B
SCHEMBL6325871 0.90 CCR3 (0.57) CCR3SSTR5HRH1HTR2B
SCHEMBL6325876 0.90 CCR3 (0.57) CCR3SSTR5HRH1HTR2B
SCHEMBL6326938 0.90 CCR3 (0.57) CCR3SSTR5HRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050090504-A1 Piperidinyl and piperazinyl compounds substituted with bicyclo-heterocyclylalkyl groups useful as CCR3 receptor antagonists ROCHE PALO ALTO LLC 2005-04-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050090504-A1 Piperidinyl and piperazinyl compounds substituted with bicyclo-heterocyclylalkyl groups useful as CCR3 receptor antagonists CCR9, CCR3, CCR1 CCR3 2/4885SSTR5 908/4885HRH1 250/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.