SCHEMBL6328150

SCHEMBL6328150

O=C(CCCc1nc(-c2cc(Cl)cc(Cl)c2)no1)NCCCCNc1n[nH]c(=O)c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.45
TSHR P16473 3/20 0.45
HPGD P15428 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP3A4 P08684 1/20 0.45
LMNA P02545 4/20 0.43
ALDH1A1 P00352 4/20 0.43
HTT P42858 2/20 0.43
MAPK1 P28482 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
USP2 O75604 1/20 0.43
TP53 P04637 1/20 0.43
AURKB Q96GD4 1/20 0.43
CNR2 P34972 1/20 0.42
HDAC1 Q13547 3/20 0.42
HDAC2 Q92769 3/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6324511 0.98 SMN1; SMN2 (0.45) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL5074272 0.96 SMN1; SMN2 (0.46) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL6330588 0.96 HPGD (0.48) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL6331242 0.94 HPGD (0.48) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL6327897 0.93 HDAC1 (0.51) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL6328068 0.91 HDAC1 (0.51) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL6332451 0.91 CYP1A2 (0.48) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL6328158 0.91 HPGD (0.53) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL6332476 0.89 NPSR1 (0.47) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6
SCHEMBL6332801 0.89 HPGD (0.53) SMN1; SMN2TSHRHPGDCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924284-B2 PARP inhibitors ICOS CORPORATION (US) 2005-08-02 US disclosed