SCHEMBL6348155

SCHEMBL6348155

O=C(O)Cc1nc(-c2nc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c3ccccc3n2)cs1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.54
ERBB2 P04626 15/20 0.54
MEN1 O00255 2/20 0.54
MAPK1 P28482 2/20 0.54
KMT2A Q03164 2/20 0.54
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP3A4 P08684 1/20 0.53
MAPT P10636 1/20 0.53
ALOX15 P16050 1/20 0.53
HSD17B10 Q99714 1/20 0.53
ERBB4 Q15303 2/20 0.52
HDAC3 O15379 2/20 0.52
ABL1 P00519 2/20 0.52
INSR P06213 2/20 0.52
PDGFRB P09619 2/20 0.52
CDK2 P24941 2/20 0.52
PLK1 P53350 2/20 0.52
HDAC4 P56524 2/20 0.52
HDAC1 Q13547 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4003729 0.85 EGFR (0.73) EGFRERBB2MEN1MAPK1KMT2A
SCHEMBL6977418 0.79 EGFR (0.75) EGFRERBB2ERBB4GAKERBB3
SCHEMBL4009625 0.73 EGFR (0.72) EGFRERBB2MEN1MAPK1KMT2A
SCHEMBL4002290 0.73 EGFR (0.62) EGFRERBB2MEN1MAPK1KMT2A
SCHEMBL28771965 0.73 EGFR (0.82) EGFRERBB2ERBB4HDAC3ABL1
SCHEMBL4003728 0.73 EGFR (0.51) EGFRERBB2MEN1MAPK1KMT2A
SCHEMBL2306317 0.72 EGFR (0.63) EGFRERBB2ERBB4HDAC3ABL1
SCHEMBL6954796 0.72 EGFR (0.84) EGFRERBB2ERBB4HDAC3ABL1
SCHEMBL6355635 0.72 EGFR (0.55) EGFRERBB2MEN1MAPK1KMT2A
SCHEMBL3702763 0.72 EGFR (0.77) EGFRERBB2ERBB4HDAC3ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6933299-B1 Anilinoquinazolines as protein tyrosine kinase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 2005-08-23 US disclosed