SCHEMBL6355265

SCHEMBL6355265

c1cn(-c2nnn[nH]2)nn1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 13/20 0.37
KEAP1 Q14145 1/20 0.33
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL218331 0.73 NOTUM (0.41) NOTUM
SCHEMBL29118314 0.72 NOTUM (0.39) NOTUM
Ammonia Solution, Strong SCHEMBL7867000 0.72 NOTUM (0.39) NOTUM
SCHEMBL28548337 0.71 NOTUM (0.49) NOTUMKEAP1CYP19A1
Ethane SCHEMBL16751833 0.71 NOTUM (0.40) NOTUM
SCHEMBL9466419 0.70 NPC1 (0.33)
SCHEMBL13407536 0.69 NOTUM (0.36) NOTUMKEAP1
Piperazine SCHEMBL7865831 0.67 NOTUM (0.35) NOTUM
SCHEMBL28456730 0.67 NOTUM (0.50) NOTUMKEAP1
Guanidine SCHEMBL7865811 0.66 MAPT (0.40) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116574068-A Universal energy-containing combustion speed catalyst, preparation method and application 西安近代化学研究所 2023-08-11 CN disclosed
US-20050272789-A1 Triazole-derived kinase inhibitors and uses thereof HALE MICHAEL R 2005-12-08 US disclosed
US-6962936-B2 Triazole-derived kinase inhibitors and uses thereof VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-11-08 US disclosed
EP-1390353-A1 TRIAZOLE-DERIVED KINASE INHIBITORS AND USES THEREOF Vertex Pharmaceuticals Incorporated (US) 2004-02-25 EP disclosed
US-20030158238-A1 Triazole-derived kinase inhibitors and uses thereof VERTEX PHARMACEUTICALS INCORPORATED 2003-08-21 US disclosed
WO-2002088097-A1 TRIAZOLE-DERIVED KINASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2002-11-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030158238-A1 Triazole-derived kinase inhibitors and uses thereof MAP3K1, MAP3K5, MAP3K19 NOTUM 3764/4885KEAP1 1370/4885CYP19A1 2050/4885
US-20050272789-A1 Triazole-derived kinase inhibitors and uses thereof MAP3K5, MAP3K1, MAP3K3 NOTUM 3626/4885KEAP1 1378/4885CYP19A1 2045/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.