SCHEMBL6355337

SCHEMBL6355337

COc1ccc(-n2c(Br)nc3c(N)ncnc32)cn1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.50
ADORA1 P30542 18/20 0.50
ADORA2B P29275 14/20 0.50
ADORA3 P0DMS8 9/20 0.50
PI4KA P42356 2/20 0.44
PI4K2B Q8TCG2 2/20 0.44
PI4K2A Q9BTU6 2/20 0.44
PI4KB Q9UBF8 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6344566 0.78 PI4KA (0.48) ADORA2AADORA1ADORA2BADORA3PI4KA
SCHEMBL30974263 0.77 ADORA2A (0.47) ADORA2AADORA1ADORA2BADORA3PI4KA
SCHEMBL27422698 0.77 ADORA2A (0.47) ADORA2AADORA1ADORA2BADORA3PI4KA
SCHEMBL6215848 0.76 PI4KA (0.51) ADORA2AADORA1ADORA2BADORA3PI4KA
SCHEMBL6354390 0.75 PI4KA (0.69) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL1755068 0.68 ADORA2A (1.00) ADORA2AADORA1ADORA2BADORA3PI4KA
SCHEMBL29439771 0.67 ADORA2A (1.00) ADORA2AADORA1ADORA2BADORA3PI4KA
SCHEMBL8832637 0.67 ADORA2A (1.00) ADORA2AADORA1ADORA2BADORA3PI4KA
SCHEMBL4142807 0.66 TLR7 (0.41) ADORA2AADORA2B
SCHEMBL10379475 0.66 ADORA2A (0.68) ADORA2AADORA1ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6841549-B1 Condensed imidazole compounds and a therapeutic agent for diabetes mellitus EISAI CO., LTD. (JP) 2005-01-11 US disclosed
EP-1221444-A1 FUSED IMIDAZOLE COMPOUNDS AND REMEDIES FOR DIABETES MELLITUS Eisai Co., Ltd. (JP) 2002-07-10 EP disclosed