SCHEMBL6356570

SCHEMBL6356570

COc1ccc2c(COC(=O)CCC(=O)O)nn(Cc3ccccc3)c2c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 2/20 0.50
PDE5A O76074 1/20 0.49
SLC22A12 Q96S37 2/20 0.43
PLA2G2A P14555 4/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
SLC16A1 P53985 1/20 0.43
MCTS1 Q9ULC4 1/20 0.43
PLA2G10 O15496 1/20 0.42
MAPT P10636 1/20 0.42
PLA2G1B P04054 1/20 0.42
ALDH1A1 P00352 3/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
LMNA P02545 1/20 0.41
CNR2 P34972 2/20 0.41
CNR1 P21554 1/20 0.40
DYRK1A Q13627 1/20 0.40
PTGER4 P35408 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5118969 0.82 PDE5A (0.71) SLC16A3PDE5APLA2G2APTGDR2SLC16A1
SCHEMBL5118966 0.77 PDE5A (0.61) PDE5APLA2G2APTGDR2MAPTPLA2G1B
SCHEMBL929883 0.74 SLC16A3 (0.74) SLC16A3SLC16A1MCTS1
SCHEMBL1120899 0.74 PDE5A (0.58) PDE5ASLC22A12PLA2G2APTGDR2PLA2G10
SCHEMBL1651401 0.73 SLC16A3 (0.62) SLC16A3PLA2G2ASLC16A1MCTS1
SCHEMBL1651049 0.72 CNR1 (0.57) SLC16A3CNR2CNR1PTGER4
SCHEMBL927453 0.72 PDE5A (0.56) SLC16A3PDE5APLA2G2APTGDR2PLA2G1B
SCHEMBL13931862 0.71 HDAC1 (0.50) PDE5APLA2G2AALDH1A1GAAPKM
SCHEMBL9321303 0.71 PTGER4 (0.59) SLC16A3PLA2G2APLA2G1BALDH1A1GAA
SCHEMBL3064842 0.71 PDE5A (0.76) PDE5APLA2G2APLA2G10MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1586572-A1 Fused pyrazolyls as anti-cancer drugs Yung Shin Pharm. Ind. Co. Ltd. (TW) 2005-10-19 EP disclosed