SCHEMBL6364173

SCHEMBL6364173

COc1ccc2cnc(Nc3cccc(Cl)c3F)nc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 1/20 0.44
EGFR P00533 8/20 0.43
FGFR1 P11362 4/20 0.43
SRC P12931 1/20 0.43
SYK P43405 1/20 0.43
ULK1 O75385 2/20 0.42
IGF1R P08069 2/20 0.41
LRRK2 Q5S007 1/20 0.40
USP2 O75604 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
PTK2 Q05397 1/20 0.39
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4921113 0.81 CSF1R (0.51) CSF1REGFRFGFR1LRRK2
SCHEMBL31590306 0.76 PIK3CA (0.46) CSF1REGFRSRCPTK2GAA
SCHEMBL20355385 0.74 EGFR (0.60) EGFRSRC
Hydrochloric Acid SCHEMBL28182076 0.74 PDGFRB (0.58) EGFRSYKUSP2LMNACYP1A2
Hydrochloric Acid SCHEMBL3757317 0.73 EGFR (0.52) CSF1REGFRIGF1R
SCHEMBL7799235 0.72 CSF1R (0.52) CSF1REGFRFGFR1SYKULK1
SCHEMBL7800417 0.72 LRRK2 (0.53) CSF1REGFRFGFR1SRCIGF1R
SCHEMBL1635586 0.71 SYK (0.51) EGFRFGFR1SRCSYKUSP2
SCHEMBL9911264 0.71 LRRK2 (0.50) EGFRSYKIGF1RLRRK2
SCHEMBL3568126 0.71 EGFR (0.69) EGFRFGFR1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050215574-A1 4-anilino quinazoline derivatives as antiproliferative agents ASTRAZENECA AB (SE) 2005-09-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050215574-A1 4-anilino quinazoline derivatives as antiproliferative agents ERBB2, ERBB4, EGFR CSF1R 1097/4885EGFR 3/4885FGFR1 42/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.