SCHEMBL6374232

SCHEMBL6374232

O=C(/C=C/c1ccc(C(F)(F)F)cc1)c1ccc(F)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 8/20 1.00
CYP1B1 Q16678 8/20 1.00
TNFRSF1A P19438 1/20 0.77
P4HB P07237 1/20 0.77
MAOB P27338 7/20 0.74
CYP1A2 P05177 1/20 0.62
MAOA P21397 1/20 0.60
CXCL12 P48061 1/20 0.58
CTSL P07711 1/20 0.57
CTSB P07858 1/20 0.57
HDAC3 O15379 1/20 0.57
ADAM17 P78536 1/20 0.57
HDAC1 Q13547 1/20 0.57
HDAC2 Q92769 1/20 0.57
HDAC10 Q969S8 1/20 0.57
HDAC11 Q96DB2 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
HDAC5 Q9UQL6 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6374235 1.00 CYP1A1 (1.00) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
SCHEMBL6200382 1.00 CYP1A1 (1.00) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
SCHEMBL6200379 1.00 CYP1A1 (1.00) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
SCHEMBL11816722 0.93 CYP1A1 (0.87) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
SCHEMBL11816718 0.93 CYP1A1 (0.87) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
Bromide SCHEMBL11817515 0.92 CYP1A1 (0.84) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
Hydrochloric Acid SCHEMBL11819369 0.92 CYP1A1 (0.84) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
Bromide SCHEMBL11817521 0.92 CYP1A1 (0.84) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
Hydrochloric Acid SCHEMBL11819375 0.92 CYP1A1 (0.84) CYP1A1CYP1B1TNFRSF1AP4HBMAOB
SCHEMBL7196521 0.88 TNFRSF1A (1.00) CYP1A1CYP1B1TNFRSF1AMAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017659-B1 SUBSTITUTED TETRAHYDRONAPHTHALINE AND ANALOGOUS COMPOUNDS BAYER HEALTHCARE AG (DE) 2005-04-27 EP disclosed
US-6586613-B1 Compounds such as 5-(tert-butyldimethylsiloxy)-7,7-dimethyl -4(4-fluorophenyl)-3-(hydroxy-(4-trifluorophenyl)-methyl)-2-isopropyl -5,6,7,8-tetrahydronaphthalene, used as antagonists for cholesteryl ester transferase protein; hyperlipemia BAYER AKTIENGELLSCHAFT (DE) 2003-07-01 US disclosed