SCHEMBL6375924

SCHEMBL6375924

CCOC(=O)c1nc2cc(-n3ccc(CNC(=O)Nc4ccccc4)c3)c(Cl)cc2[nH]c1=O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 11/20 0.54
GRIA2 P42262 11/20 0.54
GRIA3 P42263 11/20 0.54
GRIA4 P48058 11/20 0.54
GRIK1 P39086 7/20 0.49
GRIK2 Q13002 7/20 0.49
GRIK3 Q13003 7/20 0.49
GRIK4 Q16099 7/20 0.49
GRIK5 Q16478 7/20 0.49
MAPT P10636 2/20 0.42
NAMPT P43490 1/20 0.42
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6377983 0.93 GRIA1 (0.63) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6376486 0.85 GRIA1 (0.52) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6374580 0.85 GRIA1 (0.65) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6382562 0.84 GRIA1 (0.65) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6377650 0.84 GRIA1 (0.52) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6381619 0.84 GRIA1 (0.49) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6376910 0.83 GRIA1 (0.62) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6375949 0.83 GRIA1 (0.60) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6602498 0.82 GRIA1 (0.71) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL6607049 0.82 GRIA1 (0.81) GRIA1GRIA2GRIA3GRIA4GRIK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1156047-B1 6-SUBSTITUTED-7- HETEROQUINOXALINE CARBOXYLIC ACID DERIVATIVES AND ADDITION SALTS THEREOF AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN SEIYAKU KK (JP) 2005-08-31 EP disclosed
US-6632813-B1 6-subtituted-7-heteroquinoxalinecarboxylic acid derivatives and addition salts thereof and processes for the preparation of both KYORIN PHARMACEUTICAL CO., LTD. (JP) 2003-10-14 US disclosed
EP-1156047-A1 6-SUBSTITUTED-7- HETEROQUINOXALINE CARBOXYLIC ACID DERIVATIVES AND ADDITION SALTS THEREOF AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN PHARMACEUTICAL CO., LTD. (JP) 2001-11-21 EP disclosed