SCHEMBL6376259

SCHEMBL6376259

O=S(=O)(Oc1ncc(Br)cc1Cc1ccccc1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.34
NR1H3 Q13133 3/20 0.34
PTGER1 P34995 1/20 0.32
CTRC Q99895 1/20 0.32
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
DRD3 P35462 1/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
ALDH1A1 P00352 2/20 0.31
PDPK1 O15530 1/20 0.31
BCL2 P10415 1/20 0.31
BCL2L1 Q07817 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6378385 0.79 NR1H2 (0.43) NR1H2NR1H3ALDH1A1LMNA
SCHEMBL6377288 0.78 CYP11B1 (0.41) CYP11B1CYP11B2BCL2BCL2L1
SCHEMBL6377584 0.77 BCL2 (0.42) ALDH1A1BCL2LMNA
SCHEMBL6378091 0.77 NR1H2 (0.34) NR1H2NR1H3CTRCDRD2DRD1
SCHEMBL27580436 0.76 MAOB (0.41) LMNA
SCHEMBL6378848 0.74 ADORA2A (0.36) NR1H2NR1H3CYP11B1CYP11B2LMNA
SCHEMBL27580444 0.72 ADORA2A (0.36) CYP11B1CYP11B2ALDH1A1
SCHEMBL20543637 0.71 CYP11B1 (0.35) NR1H2NR1H3CYP11B1CYP11B2ALDH1A1
SCHEMBL7500214 0.70 HPGD (0.45) DRD2DRD1DRD4DRD5DRD3
SCHEMBL18583898 0.70 TAAR1 (0.53) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100334085-C Quinuclidine compound and medicine containing the same as active ingredient EISAI R & D CO LTD (JP) 2007-08-29 CN disclosed
EP-1217001-B1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT EISAI CO LTD (JP) 2005-12-07 EP disclosed
US-6599917-B1 A squalene-synthesizing enzyme inhibitor, a cholesterol biosynthesis inhibitor and a triglyceride biosynthesis inhibitor EISAI CO., LTD. (JP) 2003-07-29 US disclosed
CN-1377349-A Quinuclidine compound and medicine containing the same as active ingredient EISAI CO LTD (JP) 2002-10-30 CN disclosed
EP-1217001-A1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed