SCHEMBL6378145

SCHEMBL6378145

CC(O)C(NCCc1ccc(Cl)c(Cl)c1)Oc1ccccc1NS(C)(=O)=O

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
GRIN1 Q05586 2/20 0.43
GRIN2B Q13224 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6378590 0.84 KCNH2 (0.52) KCNH2SLC6A2SLC6A3GRIN1GRIN2B
SCHEMBL6378418 0.82 KCNH2 (0.62) KCNH2SLC6A2SLC6A3GRIN1GRIN2B
Hydrochloric Acid SCHEMBL6442762 0.82 KCNH2 (0.61) KCNH2SLC6A2SLC6A3GRIN1GRIN2B
SCHEMBL6378942 0.80 MAPT (0.43) KCNH2SLC6A2SLC6A3
SCHEMBL4206093 0.77 KCNH2 (0.71) KCNH2SLC6A2SLC6A3
SCHEMBL4216135 0.77 KCNH2 (0.71) KCNH2SLC6A2SLC6A3
SCHEMBL6379406 0.73 HSD17B10 (0.38) KCNH2
SCHEMBL6378907 0.71 KMT2A (0.43) KCNH2SLC6A2SLC6A3
SCHEMBL13948485 0.70 KCNH2 (0.59) KCNH2SLC6A2SLC6A3
SCHEMBL3405309 0.68 CYP19A1 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1436258-A4 PH-DEPENDENT NMDA RECEPTOR ANTAGONISTS UNIV EMORY (US) 2005-03-23 EP claimed
EP-1436258-A2 PH-DEPENDENT NMDA RECEPTOR ANTAGONISTS Emory University (US) 2004-07-14 EP claimed
WO-2002072542-A2 PH-DEPENDENT NMDA RECEPTOR ANTAGONISTS EMORY UNIVERSITY (US) 2002-09-19 WO claimed
EP-1436258-A4 PH-DEPENDENT NMDA RECEPTOR ANTAGONISTS UNIV EMORY (US) 2005-03-23 EP disclosed
EP-1436258-A2 PH-DEPENDENT NMDA RECEPTOR ANTAGONISTS Emory University (US) 2004-07-14 EP disclosed
WO-2002072542-A2 PH-DEPENDENT NMDA RECEPTOR ANTAGONISTS EMORY UNIVERSITY (US) 2002-09-19 WO disclosed