SCHEMBL6378792

SCHEMBL6378792

NCCNc1ccc(-c2nc3c(OC(N)=O)cccc3[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 3/20 0.54
PARP1 P09874 13/20 0.47
DHODH Q02127 5/20 0.47
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TP53 P04637 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B10 Q99714 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
PLA2G2A P14555 1/20 0.44
ALOX15 P16050 1/20 0.44
PTGS2 P35354 1/20 0.44
CHEK2 O96017 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6384304 0.89 PARP1 (0.45) HPSEPARP1DHODHTP53
SCHEMBL6384729 0.88 HPSE (0.53) HPSEPARP1DHODHKDM4ENPC1
SCHEMBL6382252 0.86 PIM1 (0.53) HPSEPARP1DHODHKDM4ENPC1
SCHEMBL6384512 0.84 PARP1 (0.56) HPSEPARP1DHODHHDAC3HDAC1
SCHEMBL6380062 0.83 PARP1 (0.44) HPSEPARP1DHODHTP53
SCHEMBL6379356 0.83 PARP1 (0.53) HPSEPARP1DHODHHDAC3HDAC1
SCHEMBL6381589 0.80 PARP1 (0.56) HPSEPARP1DHODHHDAC3HDAC1
SCHEMBL6383551 0.79 PARP1 (0.71) HPSEPARP1DHODHHDAC3HDAC1
SCHEMBL6590709 0.79 PKN1 (0.66) HPSEPARP1DHODHPARP2PLA2G2A
SCHEMBL6380064 0.78 PARP1 (0.54) HPSEPARP1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131301-B1 2-PHENYLBENZIMIDAZOLES AND 2-PHENYLINDOLES, AND PRODUCTION AND USE THEREOF ABBOTT GMBH & CO KG (DE) 2005-08-24 EP disclosed