SCHEMBL6380459

SCHEMBL6380459

COc1ccc2ncc(C#N)c(Nc3cccc(N(C)C)c3)c2c1

nearest known ligand 0.77

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.77
ERBB2 P04626 10/20 0.76
MAP2K1 Q02750 5/20 0.67
RAF1 P04049 3/20 0.67
PDE4B Q07343 1/20 0.64
SRC P12931 1/20 0.58
GAK O14976 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6382347 0.93 EGFR (0.70) EGFRERBB2MAP2K1RAF1PDE4B
Hydrochloric Acid SCHEMBL6381171 0.92 EGFR (0.70) EGFRERBB2MAP2K1RAF1PDE4B
SCHEMBL6381708 0.87 EGFR (1.00) EGFRERBB2MAP2K1RAF1SRC
SCHEMBL6381476 0.86 EGFR (0.75) EGFRERBB2MAP2K1RAF1PDE4B
SCHEMBL6381466 0.86 EGFR (0.69) EGFRERBB2MAP2K1RAF1PDE4B
SCHEMBL8143917 0.86 EGFR (0.69) EGFRERBB2MAP2K1RAF1PDE4B
SCHEMBL1893705 0.82 PDE4B (0.71) EGFRERBB2MAP2K1RAF1PDE4B
SCHEMBL6380922 0.82 PDE4B (0.71) EGFRERBB2MAP2K1RAF1PDE4B
SCHEMBL6426473 0.82 EGFR (0.66) EGFRERBB2GAK
SCHEMBL6383741 0.82 EGFR (0.63) EGFRERBB2MAP2K1RAF1PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263503-B1 USE OF CYANOQUINOLINES FOR TREATING OR INHIBITING COLONIC POLYPS WYETH CORP (US) 2005-11-02 EP claimed
EP-0973746-B1 SUBSTITUTED 3-CYANO QUINOLINES WYETH CORP (US) 2003-09-24 EP claimed