SCHEMBL6380476

SCHEMBL6380476

CN(C)Cc1cccc(-c2nc3c(OC(N)=O)cccc3[nH]2)c1

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.72
DYRK3 O43781 1/20 0.50
MAP4K4 O95819 1/20 0.50
PIM1 P11309 1/20 0.50
RPS6KB1 P23443 1/20 0.50
CSNK2A1 P68400 1/20 0.50
PKN2 Q16513 1/20 0.50
PIM3 Q86V86 1/20 0.50
BRSK1 Q8TDC3 1/20 0.50
AURKB Q96GD4 1/20 0.50
HIPK2 Q9H2X6 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
MKNK2 Q9HBH9 1/20 0.50
STK17A Q9UEE5 1/20 0.50
MAP4K5 Q9Y4K4 1/20 0.50
VSIR Q9H7M9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6381528 0.90 PARP1 (0.58) PARP1DYRK3MAP4K4PIM1RPS6KB1
SCHEMBL6379926 0.90 PARP1 (0.58) PARP1DYRK3MAP4K4PIM1RPS6KB1
SCHEMBL6381105 0.89 PARP1 (0.71) PARP1DYRK3MAP4K4PIM1RPS6KB1
SCHEMBL6383675 0.87 PARP1 (0.57) PARP1PIM1PIM3AURKBVSIR
SCHEMBL6385598 0.85 PARP1 (0.56) PARP1VSIR
SCHEMBL6380066 0.85 PARP1 (0.55) PARP1PIM1PIM3AURKBVSIR
SCHEMBL6383270 0.84 PARP1 (0.51) PARP1DYRK3MAP4K4PIM1RPS6KB1
SCHEMBL7134234 0.84 PARP1 (1.00) PARP1DYRK3MAP4K4PIM1RPS6KB1
SCHEMBL6378984 0.83 PARP1 (0.51) PARP1VSIR
SCHEMBL6579124 0.82 MAP4K4 (0.75) PARP1DYRK3MAP4K4PIM1RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131301-B1 2-PHENYLBENZIMIDAZOLES AND 2-PHENYLINDOLES, AND PRODUCTION AND USE THEREOF ABBOTT GMBH & CO KG (DE) 2005-08-24 EP disclosed