SCHEMBL6409195

SCHEMBL6409195

Nc1ccc2c(c1)C(=Cc1ccc3[nH]ccc3c1)C(=O)N2

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RET P07949 7/20 0.58
ALK Q9UM73 4/20 0.57
FLT3 P36888 2/20 0.57
PDPK1 O15530 1/20 0.57
RPS6KA3 P51812 1/20 0.50
PIM1 P11309 1/20 0.46
CYP2A6 P11509 1/20 0.44
PLK4 O00444 1/20 0.44
LRRK2 Q5S007 2/20 0.43
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
CHEK1 O14757 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6409193 1.00 RET (0.58) RETALKFLT3PDPK1RPS6KA3
SCHEMBL5182063 0.84 PDPK1 (0.60) PDPK1
SCHEMBL5182059 0.84 PDPK1 (0.60) PDPK1
SCHEMBL5473028 0.84 PDGFRB (0.57) RETALKFLT3PDPK1RPS6KA3
SCHEMBL5473025 0.84 PDGFRB (0.57) RETALKFLT3PDPK1RPS6KA3
SCHEMBL6409208 0.82 TLK2 (0.60) PDPK1PIM1
SCHEMBL6409203 0.82 TLK2 (0.60) PDPK1PIM1
SCHEMBL5843095 0.81 PDPK1 (0.47) PDPK1PLK4LRRK2PSEN1PSEN2
SCHEMBL5843099 0.81 PDPK1 (0.47) PDPK1PLK4LRRK2PSEN1PSEN2
SCHEMBL5430411 0.79 CDK2 (0.52) PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855730-B2 3-methylidenyl-2-indolinone modulators of protein kinase SUGEN, INC. (US) 2005-02-15 US disclosed
US-20040024010-A1 3-methylidenyl-2-indolinone modulators of protein kinase SUGEN, INC. 2004-02-05 US disclosed
US-6531502-B1 Antitumor SUGEN, INC. 2003-03-11 US disclosed
WO-2000008202-A9 3-METHYLIDENYL-2-INDOLINONE MODULATORS OF PROTEIN KINASE SUGEN INC (US) 2000-07-27 WO disclosed
WO-2000008202-A2 3-METHYLIDENYL-2-INDOLINONE MODULATORS OF PROTEIN KINASE SUGEN, INC. (US) 2000-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040024010-A1 3-methylidenyl-2-indolinone modulators of protein kinase DMPK, MAP4K3, MAP3K20 RET 487/4885ALK 1033/4885FLT3 812/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.