SCHEMBL6422356

SCHEMBL6422356

Nc1ccc(N2CCC3(CCCC(=O)N3Cc3cccc4[nH]ccc34)CC2)nc1

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 20/20 0.72
HCRTR1 O43613 18/20 0.72
KCNH2 Q12809 1/20 0.44
LTC4S Q16873 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2130816 0.87 HCRTR1 (0.69) HCRTR2HCRTR1KCNH2LTC4S
SCHEMBL2025800 0.83 HCRTR1 (1.00) HCRTR2HCRTR1KCNH2LTC4S
SCHEMBL2136234 0.82 HCRTR2 (0.73) HCRTR2HCRTR1KCNH2LTC4S
SCHEMBL2135877 0.82 HCRTR2 (0.74) HCRTR2HCRTR1KCNH2LTC4S
SCHEMBL12700416 0.81 HCRTR1 (0.61) HCRTR2HCRTR1KCNH2
SCHEMBL2132818 0.80 HCRTR1 (0.68) HCRTR2HCRTR1KCNH2LTC4S
SCHEMBL2133982 0.80 HCRTR1 (0.65) HCRTR2HCRTR1KCNH2LTC4S
SCHEMBL2130371 0.80 HCRTR2 (0.70) HCRTR2HCRTR1KCNH2LTC4S
SCHEMBL2136120 0.79 HCRTR1 (1.00) HCRTR2HCRTR1
SCHEMBL2130316 0.78 HCRTR1 (0.82) HCRTR2HCRTR1KCNH2LTC4S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012055888-A1 DIAZA-SPIRO[5.5]UNDECANES USEFUL AS OREXIN RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2012-05-03 WO disclosed