SCHEMBL6428028

SCHEMBL6428028

[CH2]c1cc(C#Cc2ccc(-c3ccc(Cl)cc3)cn2)ccc1OCCN1CCCC1

nearest known ligand 0.82

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 20/20 0.82
CHRM1 P11229 4/20 0.73
HTR2A P28223 3/20 0.73
CYP2D6 P10635 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2323784 0.90 MCHR1 (1.00) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL13920752 0.89 MCHR1 (0.79) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2319702 0.88 MCHR1 (0.82) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2322221 0.88 MCHR1 (0.82) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2321296 0.88 MCHR1 (0.82) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2327427 0.88 MCHR1 (0.82) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4485373 0.88 MCHR1 (0.82) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2323051 0.88 MCHR1 (0.82) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2322440 0.87 MCHR1 (0.80) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2328524 0.87 MCHR1 (0.80) MCHR1CHRM1HTR2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558578-A1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2005-08-03 EP disclosed
WO-2004039780-A1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-05-13 WO disclosed