SCHEMBL6433437

SCHEMBL6433437

O=C(O)C[C@H](c1cccc(F)c1)N1CCN(CCCc2ccc3c(n2)NCCC3)C1=O

nearest known ligand 0.82

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.82
ITGB6 P18564 7/20 0.82
ITGB8 P26012 4/20 0.82
ITGB3 P05106 18/20 0.78
ITGA2B P08514 4/20 0.68
ITGB1 P05556 1/20 0.68
ITGA5 P08648 1/20 0.68
ITGB5 P18084 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6432131 1.00 ITGAV (0.82) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL6432134 1.00 ITGAV (0.82) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL25665881 0.91 ITGAV (0.80) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL17999152 0.90 ITGAV (1.00) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL17999154 0.90 ITGAV (1.00) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL29707555 0.90 ITGAV (1.00) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL22209127 0.89 ITGAV (0.81) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL22209130 0.89 ITGAV (0.81) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL22223362 0.89 ITGAV (0.81) ITGAVITGB6ITGB8ITGB3ITGA2B
SCHEMBL6432148 0.88 ITGAV (0.78) ITGAVITGB6ITGB8ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040111-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-06-22 EP claimed
EP-1040111-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-06-22 EP disclosed
US-6017926-A Integrin receptor antagonists MERCK & CO., INC. (US) 2000-01-25 US disclosed