SCHEMBL6433503

SCHEMBL6433503

Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CN(C(CO)C(O)CBr)C1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.61
LCK P06239 4/20 0.61
LYN P07948 1/20 0.61
NUDT14 O95848 1/20 0.58
NUDT5 Q9UKK9 1/20 0.58
SRC P12931 1/20 0.55
KDR P35968 1/20 0.55
TEK Q02763 1/20 0.55
BLK P51451 1/20 0.54
EGFR P00533 3/20 0.54
ITK Q08881 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6434459 0.83 BTK (0.66) BTKLCKLYNNUDT14NUDT5
SCHEMBL6431810 0.83 BTK (0.66) BTKLCKLYNNUDT14NUDT5
SCHEMBL25068919 0.82 BTK (0.73) BTKLCKLYNNUDT14NUDT5
2-Bromoethanol SCHEMBL6433498 0.81 BTK (0.66) BTKLCKLYNNUDT14NUDT5
SCHEMBL5803152 0.81 BTK (0.70) BTKLCKLYNNUDT14NUDT5
SCHEMBL27586609 0.80 BTK (0.67) BTKLCKLYNNUDT14NUDT5
SCHEMBL24196789 0.79 BTK (0.81) BTKLCKLYNNUDT14NUDT5
SCHEMBL5817900 0.79 BTK (0.73) BTKLCKLYNNUDT14NUDT5
SCHEMBL7144296 0.79 BTK (0.73) BTKLCKLYNNUDT14NUDT5
SCHEMBL27586611 0.78 BTK (0.67) BTKLCKLYNNUDT14NUDT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6921763-B2 Pyrazolopyrimidines as therapeutic agents ABBOTT LABORATORIES (US) 2005-07-26 US disclosed
US-6660744-B1 Kinase inhibitors ABBOTT GMBH & CO. KG (DE) 2003-12-09 US disclosed
EP-1212327-B1 PYRAZOLOPYRIMIDINES AS THERAPEUTIC AGENTS BASF AG (DE) 2003-08-20 EP disclosed