SCHEMBL6433880

SCHEMBL6433880

COc1cc2c(Nc3cc(O)c(Cl)cc3F)ccnc2cc1OCc1ccncc1

nearest known ligand 0.75

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 7/20 0.75
FGFR1 P11362 5/20 0.75
KDR P35968 12/20 0.58
FLT4 P35916 2/20 0.57
FGFR2 P21802 1/20 0.57
FGFR4 P22455 1/20 0.57
FGFR3 P22607 1/20 0.57
EGFR P00533 4/20 0.53
SRC P12931 2/20 0.52
ERBB2 P04626 1/20 0.52
EPHA2 P29317 1/20 0.52
RET P07949 4/20 0.47
KIF5B P33176 4/20 0.47
RAF1 P04049 2/20 0.47
BRAF P15056 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6430947 0.99 FLT1 (0.74) FLT1FGFR1KDRFLT4FGFR2
SCHEMBL6430998 0.93 FLT1 (0.75) FLT1FGFR1KDRFLT4FGFR2
Hydrochloric Acid SCHEMBL6431427 0.92 FLT1 (0.74) FLT1FGFR1KDRFLT4FGFR2
SCHEMBL6437903 0.89 FLT1 (0.84) FLT1FGFR1KDRFLT4FGFR2
SCHEMBL6095959 0.88 KDR (0.73) FLT1FGFR1KDRFLT4FGFR2
Hydrochloric Acid SCHEMBL6435465 0.88 FLT1 (0.83) FLT1FGFR1KDRFLT4FGFR2
SCHEMBL7458759 0.88 KDR (0.75) FLT1FGFR1KDRFLT4FGFR2
SCHEMBL6436401 0.88 FLT1 (0.82) FLT1FGFR1KDRFLT4FGFR2
Hydrochloric Acid SCHEMBL7459204 0.87 KDR (0.74) FLT1FGFR1KDRFLT4FGFR2
Hydrochloric Acid SCHEMBL6431121 0.87 FLT1 (0.80) FLT1FGFR1KDRFLT4FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP claimed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US claimed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP claimed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO claimed
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed