SCHEMBL6433988

SCHEMBL6433988

COCCOc1cc2nccc(Oc3cccc(O)c3)c2cc1C#N

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 2/20 0.47
CSF1R P07333 1/20 0.47
FLT4 P35916 1/20 0.47
FLT3 P36888 1/20 0.47
EGFR P00533 4/20 0.46
ERBB2 P04626 2/20 0.43
KDR P35968 3/20 0.43
MET P08581 2/20 0.43
AURKA O14965 2/20 0.43
LCK P06239 2/20 0.43
TEK Q02763 2/20 0.43
FLT1 P17948 2/20 0.43
LYN P07948 1/20 0.43
AURKB Q96GD4 1/20 0.43
AXL P30530 1/20 0.43
RET P07949 1/20 0.43
KIF5B P33176 1/20 0.43
PDGFRA P16234 1/20 0.42
FGFR1 P11362 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1895568 0.84 PDGFRA (0.58) PDGFRBCSF1RFLT4FLT3KDR
SCHEMBL1891081 0.82 AXL (0.47) PDGFRBCSF1RFLT4FLT3KDR
SCHEMBL1896916 0.80 PDGFRA (0.58) KDRMETAXLPDGFRA
SCHEMBL1895977 0.80 AXL (0.45) PDGFRBCSF1RFLT4FLT3KDR
SCHEMBL1894126 0.80 PDGFRB (0.43) PDGFRBCSF1RFLT4FLT3KDR
SCHEMBL12501727 0.80 AXL (0.47) PDGFRBCSF1RFLT4FLT3KDR
SCHEMBL1889956 0.79 PDGFRB (0.43) PDGFRBCSF1RFLT4FLT3KDR
SCHEMBL14540580 0.79 AXL (0.52) PDGFRBCSF1RFLT4FLT3KDR
SCHEMBL1896541 0.79 PDGFRA (0.70) PDGFRBCSF1RFLT4FLT3KDR
SCHEMBL4338322 0.79 AXL (0.59) PDGFRBCSF1RFLT4FLT3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed