SCHEMBL6437693

SCHEMBL6437693

COOC(=O)C(OC)(c1ccccc1)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.44
CES1 P23141 1/20 0.41
NR1H2 P55055 2/20 0.39
NR1H3 Q13133 2/20 0.39
MAPK1 P28482 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ENPP2 Q13822 2/20 0.37
GAA P10253 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
VEGFA P15692 1/20 0.36
ALDH1A1 P00352 4/20 0.35
PTPN1 P18031 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 4/20 0.34
SRC P12931 1/20 0.34
LMNA P02545 3/20 0.34
APAF1 O14727 1/20 0.34
TDP2 O95551 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8171410 0.86 KCNN4 (0.56) KCNN4CES1NR1H2NR1H3MAPK1
SCHEMBL27910386 0.86 KCNN4 (0.47) KCNN4CES1NR1H2NR1H3MAPK1
SCHEMBL236357 0.84 CES1 (0.47) KCNN4CES1NR1H2NR1H3MAPK1
SCHEMBL246914 0.84 CES1 (0.47) KCNN4CES1NR1H2NR1H3MAPK1
SCHEMBL236358 0.84 CES1 (0.47) KCNN4CES1NR1H2NR1H3MAPK1
Hydrochloric Acid SCHEMBL4926039 0.82 CES1 (0.46) KCNN4CES1NR1H2NR1H3MAPK1
Hydrochloric Acid SCHEMBL5595770 0.82 CES1 (0.46) KCNN4CES1NR1H2NR1H3MAPK1
Hydrochloric Acid SCHEMBL8829227 0.82 CES1 (0.46) KCNN4CES1NR1H2NR1H3MAPK1
SCHEMBL27910400 0.82 KCNN4 (0.43) KCNN4CES1NR1H2NR1H3MAPK1
SCHEMBL12712220 0.82 KCNN4 (0.43) KCNN4CES1NR1H2NR1H3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1513527-A1 PRODRUGS OF IMIDAZOLE DERIVATIVES, FOR USE AS PROTON PUMP INHIBITORS IN THE TREATMENT OF E.G. PEPTIC ULCERS Takeda Pharmaceutical Company Limited (JP) 2005-03-16 EP disclosed
WO-2003105845-A1 PRODRUGS OF IMIDAZOLE DERIVATIVES, FOR USE AS PROTON PUMP INHIBITORS IN THE TREATMENT OF E.G. PEPTIC ULCERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-12-24 WO disclosed