SCHEMBL6440111

SCHEMBL6440111

CCCc1cc(C(CC)(CC)c2cc(C)c(C(=O)OC)s2)ccc1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.44
ESR2 Q92731 9/20 0.44
AR P10275 3/20 0.40
HDAC3 O15379 2/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HPGD P15428 2/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
CYP2C19 P33261 1/20 0.36
CKS1B P61024 1/20 0.36
SKP2 Q13309 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36
VDR P11473 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393109 0.88 ESR1 (0.53) ESR1ESR2ARHDAC3HDAC6
SCHEMBL3392386 0.82 ESR1 (0.40) ESR1ESR2ARHDAC3HDAC6
SCHEMBL3394907 0.82 HPGD (0.52) ESR1ESR2ARHPGDALDH1A1
SCHEMBL13366689 0.78 ESR1 (0.48) ESR1HDAC3HDAC6VDR
SCHEMBL13672861 0.77 HDAC3 (0.37) ESR1ESR2ARHDAC3HDAC6
SCHEMBL13366680 0.77 HDAC3 (0.43) HDAC3HDAC6HPGDALDH1A1VDR
SCHEMBL3393336 0.77 HDAC3 (0.54) ARHDAC3HDAC6VDRL3MBTL1
SCHEMBL3391173 0.75 HDAC3 (0.58) ESR1ARHDAC3HDAC6VDR
SCHEMBL3388734 0.75 HDAC6 (0.45) HDAC3HDAC6HPGDVDRL3MBTL1
SCHEMBL3396335 0.74 ESR1 (0.57) ESR1ESR2ARVDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511740-A1 PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2005-03-09 EP disclosed
WO-2003101978-A1 PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2003-12-11 WO disclosed