SCHEMBL6440199

SCHEMBL6440199

Oc1ccc(-n2c(C3CCCC3)nc3ccccc32)cc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 5/20 0.54
ESR1 P03372 4/20 0.54
SCN9A Q15858 3/20 0.52
GRIA1 P42261 1/20 0.49
CACNG8 Q8WXS5 1/20 0.49
CACNG2 Q9Y698 1/20 0.49
USP2 O75604 1/20 0.48
POLB P06746 1/20 0.48
CNR2 P34972 6/20 0.46
CNR1 P21554 2/20 0.45
CYP1A2 P05177 1/20 0.43
PDE10A Q9Y233 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6916575 1.00 ESR2 (0.54) ESR2ESR1SCN9AGRIA1CACNG8
SCHEMBL6461068 0.97 ESR2 (0.54) ESR2ESR1SCN9AGRIA1CACNG8
SCHEMBL6439085 0.94 ESR2 (0.56) ESR2ESR1SCN9AGRIA1CACNG8
SCHEMBL8022188 0.87 USP2 (0.54) SCN9AUSP2POLBCNR2CNR1
SCHEMBL10818327 0.82 SCN9A (0.55) SCN9AUSP2POLBCYP1A2PDE10A
SCHEMBL6439386 0.81 ESR2 (0.62) ESR2ESR1SCN9AGRIA1CACNG8
SCHEMBL13052920 0.79 USP2 (0.52) SCN9AUSP2POLBCNR2CNR1
SCHEMBL7887660 0.75 SCN9A (0.50) SCN9ACYP1A2PDE10A
SCHEMBL18334017 0.75 MAPK10 (0.46) SCN9AUSP2POLBCNR2CNR1
SCHEMBL6440718 0.73 ESR2 (0.52) ESR2ESR1SCN9AGRIA1CACNG8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517897-A2 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS ESTROGEN AGONISTS/ANTAGONISTS Pfizer Products Inc. (US) 2005-03-30 EP disclosed
WO-2004000817-A2 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS ESTROGEN AGONISTS/ANTAGONISTS PFIZER PRODUCTS INC. (US) 2003-12-31 WO disclosed