SCHEMBL6441209

SCHEMBL6441209

CNC(=O)Oc1cccc2c(C(=O)C(=O)N3CCN(C(=O)c4ccccc4)C[C@H]3C)c[nH]c12

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 6/20 0.66
CYP2D6 P10635 5/20 0.66
CYP2C9 P11712 5/20 0.66
CYP3A4 P08684 3/20 0.58
GABRA1 P14867 2/20 0.42
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42
GABRA3 P34903 2/20 0.42
GABRA2 P47869 2/20 0.42
GABRB2 P47870 2/20 0.42
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GHSR Q92847 2/20 0.39
SMO Q99835 3/20 0.37
ALOX5 P09917 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C8 P10632 1/20 0.37
CYP2B6 P20813 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6444155 0.91 CYP2C19 (0.63) CYP2C19CYP2D6CYP2C9CYP3A4GABRA1
SCHEMBL6441753 0.90 CYP2C19 (0.66) CYP2C19CYP2D6CYP2C9CYP3A4GABRA1
SCHEMBL6442331 0.86 CYP2C19 (0.57) CYP2C19CYP2D6CYP2C9CYP3A4GABRA1
SCHEMBL6445271 0.86 CYP2C19 (0.70) CYP2C19CYP2D6CYP2C9CYP3A4GABRA1
SCHEMBL6445265 0.86 CYP2C19 (0.70) CYP2C19CYP2D6CYP2C9CYP3A4GABRA1
SCHEMBL6441344 0.84 CYP2C19 (0.70) CYP2C19CYP2D6CYP2C9CYP3A4GABRA1
SCHEMBL6441347 0.84 CYP2C19 (0.70) CYP2C19CYP2D6CYP2C9CYP3A4GABRA1
SCHEMBL6442492 0.84 CYP2C19 (0.75) CYP2C19CYP2D6CYP2C9CYP3A4HTT
SCHEMBL6442498 0.84 CYP2C19 (0.75) CYP2C19CYP2D6CYP2C9CYP3A4HTT
SCHEMBL11963655 0.84 CYP2C19 (0.67) CYP2C19CYP2D6CYP2C9CYP3A4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299382-B1 COMPOSITION AND ANTIVIRAL ACTIVITY OF SUBSTITUTED INDOLEOXOACETIC PIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2005-09-21 EP claimed