SCHEMBL6445667

SCHEMBL6445667

COc1cccc(C(=O)CN2c3nc(-c4ccncc4)cc(=O)n3CCC2c2ccccc2)c1.COc1ccccc1C(=O)CN1c2nc(-c3ccncc3)cc(=O)n2CCC1c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 12/20 0.42
CYP2D6 P10635 3/20 0.42
MAPT P10636 2/20 0.37
PRKACA P17612 1/20 0.37
ROCK1 Q13464 1/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KDR P35968 1/20 0.36
ALDH1A1 P00352 1/20 0.36
THRB P10828 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315291 0.94 GSK3B (0.47) GSK3BCYP2D6MAPTPRKACAROCK1
SCHEMBL315955 0.93 GSK3B (0.43) GSK3BCYP2D6MAPTALDH1A1CYP1A2
SCHEMBL316072 0.86 GSK3B (0.44) GSK3BCYP2D6MAPTL3MBTL1ALDH1A1
Hydrochloric Acid SCHEMBL315968 0.85 GSK3B (0.45) GSK3BCYP2D6MAPTL3MBTL1ALDH1A1
SCHEMBL315314 0.84 GSK3B (0.46) GSK3BCYP2D6TDP1ALDH1A1CYP1A2
SCHEMBL315639 0.84 GSK3B (0.46) GSK3BCYP2D6TDP1ALDH1A1CYP1A2
SCHEMBL4865807 0.84 GSK3B (0.45) GSK3BCYP2D6MAPTMAPK1ALDH1A1
Hydrochloric Acid SCHEMBL315474 0.83 GSK3B (0.46) GSK3BCYP2D6TDP1ALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL315489 0.83 GSK3B (0.46) GSK3BCYP2D6TDP1ALDH1A1CYP1A2
SCHEMBL317015 0.82 GSK3B (0.49) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608654-A2 8-SUBSTITUTED-6, 7, 8,9-TETRAHY9DROPYRIMIDO (1,2- a) PYRIMIDIN-4-ONE DERIVATIVES Sanofi-Aventis (FR) 2005-12-28 EP claimed
WO-2004082577-A2 8-SUBSTITUTED-6, 7, 8, 9-TETRAHYDROPYRIMIDO[1,2-a] PYRIMIDIN-4-ONE DERIVATIVES SANOFI-AVENTIS (FR) 2004-09-30 WO claimed