SCHEMBL644635

SCHEMBL644635

COc1ccccc1CN(C)S(=O)(=O)c1cc(-c2nnc(O)n2-c2ccccc2F)c(O)cc1O

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 6/20 0.51
HSP90AB1 P08238 1/20 0.42
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAOB P27338 2/20 0.35
KMT2A Q03164 1/20 0.35
KCNN4 O15554 1/20 0.34
MAOA P21397 1/20 0.34
CASP3 P42574 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL646628 0.96 HSP90AA1 (0.51) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2KMT2A
SCHEMBL647531 0.93 HSP90AA1 (0.49) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2KMT2A
SCHEMBL645831 0.92 HSP90AA1 (0.51) HSP90AA1HSP90AB1MAOBKMT2A
SCHEMBL646679 0.92 HSP90AA1 (0.55) HSP90AA1HSP90AB1MAOBMAOACASP3
SCHEMBL647555 0.91 HSP90AA1 (0.49) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2KMT2A
SCHEMBL645378 0.91 HSP90AA1 (0.48) HSP90AA1HSP90AB1MAOBKMT2AKCNN4
SCHEMBL645400 0.91 HSP90AA1 (0.48) HSP90AA1HSP90AB1MAOBKCNN4MAOA
SCHEMBL646699 0.90 HSP90AA1 (0.49) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2MAOB
SCHEMBL645488 0.90 HSP90AA1 (0.51) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2KMT2A
SCHEMBL10179897 0.90 HSP90AA1 (0.49) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2023922-B1 TRIAZOLE DERIVATIVES II MERCK PATENT GMBH (DE) 2012-07-11 EP claimed
US-8119795-B2 Triazole derivatives II MERCK PATENT GMBH (DE) 2012-02-21 US claimed
US-20100022540-A1 TRIAZOLE DERIVATIVES II MERCK PATENT GESELLSCHAFT (DE) 2010-01-28 US claimed
EP-2023922-B1 TRIAZOLE DERIVATIVES II MERCK PATENT GMBH (DE) 2012-07-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100022540-A1 TRIAZOLE DERIVATIVES II HSP90AB1, HSP90AA1, HSP90AB2P HSP90AA1 2/4885HSP90AB1 1/4885ALDH1A1 1671/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.