SCHEMBL6448844

SCHEMBL6448844

[CH2]C(Cc1cccc2ccccc12)CN(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.51
CYP1A2 P05177 3/20 0.51
CYP2C19 P33261 3/20 0.51
CTNNB1 P35222 1/20 0.43
MMP9 P14780 1/20 0.43
LMNA P02545 4/20 0.42
MAPK1 P28482 2/20 0.42
ALDH1A1 P00352 1/20 0.42
NPY1R P25929 1/20 0.42
NPY2R P49146 1/20 0.42
CYP2C9 P11712 1/20 0.42
SIGMAR1 Q99720 3/20 0.40
NR1I2 O75469 2/20 0.39
SLC6A2 P23975 2/20 0.39
HTR2A P28223 2/20 0.39
SLC6A4 P31645 2/20 0.39
KCNH2 Q12809 2/20 0.39
ADRA2C P18825 2/20 0.39
ADRA1A P35348 2/20 0.39
ADRA2A P08913 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445467 0.81 HTR1B (0.47) CYP2D6CYP1A2CYP2C19CTNNB1MMP9
SCHEMBL6444377 0.78 CTNNB1 (0.46) CYP2D6CYP1A2CYP2C19CTNNB1MMP9
SCHEMBL4817621 0.77 CYP1A2 (0.50) CYP2D6CYP1A2CYP2C19CTNNB1CYP2C9
SCHEMBL9666915 0.76 CYP2D6 (0.47) CYP2D6CYP1A2CYP2C19CTNNB1MMP9
SCHEMBL9666926 0.76 CYP1A2 (0.47) CYP2D6CYP1A2CYP2C19CTNNB1MMP9
SCHEMBL6444646 0.74 CTNNB1 (0.51) CYP2D6CYP1A2CYP2C19CTNNB1MMP9
SCHEMBL6448972 0.73 CTNNB1 (0.43) CYP2D6CYP1A2CYP2C19CTNNB1LMNA
SCHEMBL6445099 0.73 CTNNB1 (0.53) CYP2D6CYP1A2CYP2C19CTNNB1CYP2C9
SCHEMBL7528890 0.72 CYP1A2 (0.53) CYP2D6CYP1A2CYP2C19CTNNB1CYP2C9
SCHEMBL31316173 0.72 CYP2D6 (0.77) CYP2D6CYP1A2CYP2C19LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050130941-A1 Methods of treating alzheimer's disease PHARMACIA & UPJOHN COMPANY LLC 2005-06-16 US disclosed
EP-1392315-A1 METHODS OF TREATING ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2004-03-03 EP disclosed
WO-2002100410-A1 METHODS OF TREATING ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed
US-5753652-A Antiretroviral hydrazine derivatives NOVARTIS CORPORATION (US) 1998-05-19 US disclosed
EP-0521827-B1 Pharmacological active hydrazin derivatives and process for their preparation CIBA GEIGY AG (CH) 1996-09-25 EP disclosed
EP-0521827-A1 Pharmacological active hydrazin derivatives and process for their preparation CIBA-GEIGY AG (CH) 1993-01-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050130941-A1 Methods of treating alzheimer's disease BACE1, PSEN1, BACE2 CYP2D6 3661/4885CYP1A2 1864/4885CYP2C19 1268/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.