SCHEMBL6449270

SCHEMBL6449270

O=C(CCc1cnn2c(=O)nc[nH]c12)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
MAPT P10636 1/20 0.37
POLB P06746 1/20 0.37
TOP2A P11388 1/20 0.37
BRAF P15056 1/20 0.37
NPY5R Q15761 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NFKB1 P19838 1/20 0.36
ALDH1A1 P00352 3/20 0.36
HSD17B10 Q99714 1/20 0.36
GLA P06280 1/20 0.36
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
GPR35 Q9HC97 1/20 0.35
GAA P10253 1/20 0.35
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4173932 0.91 MAPT (0.35) MAPTNPY5RALDH1A1GLAROCK2
SCHEMBL4158592 0.78 CYP2C9 (0.38) CYP1A2CYP2C9MAPTPOLBNPY5R
SCHEMBL4173946 0.74 MAPT (0.35) MAPTNPY5RMEN1KMT2AALDH1A1
SCHEMBL4173277 0.72 HPGD (0.31) HSD17B10HPGDTSHR
SCHEMBL4160554 0.72 PARP1 (0.36) CYP2C9MAPTPOLBNPY5RMEN1
SCHEMBL4175164 0.71 RECQL (0.39) MAPTPOLBMEN1KMT2AALDH1A1
SCHEMBL4170513 0.71 SMN1; SMN2 (0.35) MAPTPOLBNPY5RALDH1A1GLA
Leteprinim SCHEMBL358492 0.70 HSD17B10 (0.42) CYP1A2CYP2C9MAPTPOLBMEN1
SCHEMBL4158588 0.69 MAPT (0.37) MAPTMEN1KMT2AALDH1A1GLA
SCHEMBL4836350 0.68 CYP2C9 (0.46) CYP1A2CYP2C9MAPTPOLBNPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1525205-A2 NOVEL SUBSTITUTED PYRAZOLO( 1,5-A /I ]-1,3,5-TRIAZINE DERIVATIVES AND THEIR ANALOGUES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME, USE THEREOF AS MEDICINE AND METHODS FOR PREPARING SAME Greenpharma (FR) 2005-04-27 EP disclosed
WO-2004011464-A2 NOVEL SUBSTITUTED PYRAZOLO[1,5 A]-1,3,5-TRIAZINE DERIVATIVES AND THEIR ANALOGUES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME, USE THEREOF AS MEDICINE AND METHODS FOR PREPARING SAME GREENPHARMA (FR) 2004-02-05 WO disclosed