SCHEMBL6449882

SCHEMBL6449882

COC(C(=O)NCc1ccc(C(=N)N)cc1)c1c(F)ccc(C(=O)N2CCOCC2)c1F

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
ST14 Q9Y5Y6 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
F2 P00734 8/20 0.37
F10 P00742 1/20 0.37
TPSAB1 Q15661 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37
TPSD1 Q9BZJ3 1/20 0.37
TPSG1 Q9NRR2 1/20 0.37
TSHR P16473 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
TMPRSS11D O60235 1/20 0.36
MASP2 O00187 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6449886 1.00 KMT2A (0.40) KMT2AST14NOS3NOS1F2
Acetic Acid SCHEMBL5037910 0.98 F2 (0.41) KMT2AST14NOS3NOS1F2
SCHEMBL5047158 0.91 KMT2A (0.39) KMT2AKDM4EMAPTTSHRALDH1A1
SCHEMBL5047161 0.91 KMT2A (0.39) KMT2AKDM4EMAPTTSHRALDH1A1
Acetic Acid SCHEMBL5042954 0.79 ST14 (0.41) ST14F2F10TPSAB1PRSS1
Acetic Acid SCHEMBL5038366 0.78 ST14 (0.41) ST14F2F10TPSAB1PRSS1
Acetic Acid SCHEMBL5047897 0.78 ST14 (0.39) ST14F2F10PRSS1MASP2
SCHEMBL6448878 0.77 ST14 (0.50) ST14F2F10TPSAB1PRSS1
SCHEMBL6448875 0.77 ST14 (0.50) ST14F2F10TPSAB1PRSS1
Acetic Acid SCHEMBL5037784 0.77 F2 (0.42) ST14F2TPSAB1PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-08-31 EP disclosed
WO-2004048335-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-06-10 WO disclosed